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Somatostatin CAS:51110-01-1
Somatostatin ndi mahomoni achilengedwe omwe amaletsa kutulutsidwa kwa mahomoni ena osiyanasiyana m'thupi. Amagwira ntchito yofunika kwambiri pakulamulira dongosolo la endocrine ndipo amagwira ntchito yolamulira kukula kwa mahomoni, insulin, glucagon, ndi mahomoni ena am'mimba.
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Linaclotide CAS: 851199-59-2
Linaclotide ndi mankhwala a guanylate cyclase-C omwe amagwiritsidwa ntchito pochiza kudzimbidwa kosatha komanso matenda a m'mimba omwe amayambitsidwa ndi kudzimbidwa mwa akuluakulu. Amagwira ntchito m'mimba kuti awonjezere kutulutsa kwamadzimadzi ndikufulumizitsa kutuluka kwa matumbo, kuchepetsa zizindikiro zokhudzana ndi matendawa.
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Levosimendan CAS:141505-33-1
Levosimendan ndi mankhwala otsegula njira ya calcium yomwe imagwiritsidwa ntchito pochiza kulephera kwa mtima komwe kwachepa. Mankhwalawa ali ndi mphamvu zochepetsera kutentha kwa thupi komanso zotumphukira m'magazi, kukonza magwiridwe antchito a mtima ndikuchepetsa zizindikiro za kulephera kwa mtima.
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Liraglutide CAS:204656-20-2
Liraglutide ndi mankhwala omwe amagwiritsidwa ntchito pochiza matenda a shuga amtundu wachiwiri komanso kunenepa kwambiri. Ndi m'gulu la mankhwala omwe amadziwika kuti glucagon-like peptide-1 (GLP-1) receptor agonists, omwe amagwira ntchito powonjezera kupanga insulin ndikuchepetsa kuchuluka kwa shuga wopangidwa ndi chiwindi. Liraglutide imapezeka mu jakisoni ndipo nthawi zambiri imaperekedwa kamodzi patsiku. Mankhwalawa awonetsedwa kuti amathandiza kuchepetsa shuga m'magazi ndikuchepetsa thupi mwa anthu omwe ali ndi matenda a shuga amtundu wachiwiri komanso kunenepa kwambiri.
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Octreotide Acetate CAS: 83150-76-9
Octreotide acetate ndi octapeptide yopangidwa ndi mahomoni achilengedwe otchedwa somatostatin. Imagwira ntchito ngati choletsa champhamvu cha mahomoni osiyanasiyana ndi ma neuropeptides, ndipo imagwiritsidwa ntchito pochiza matenda monga acromegaly, carcinoid syndrome, ndi mitundu ina ya zotupa.
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Semaglutide CAS:910463-68-2
Semaglutide ndi glucagon-like peptide-1 (GLP-1) receptor agonist yomwe imagwiritsidwa ntchito pochiza matenda a shuga amtundu wa 2 komanso kunenepa kwambiri. Imagwira ntchito poletsa kuchuluka kwa shuga m'magazi, kuchepetsa thupi, komanso kuchepetsa chiopsezo cha matenda a mtima.
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Icatibant Acetate CAS:138614-30-9
Icatibant acetate ndi mankhwala omwe amagwiritsidwa ntchito pochiza angioedema yobadwa nayo (HAE), matenda osowa kwambiri omwe amadziwika ndi kutupa kwadzidzidzi komanso koopsa kwa khungu, nembanemba ya mucous, ndi minofu ina ya thupi. Ndi mankhwala osankhidwa a bradykinin B2 receptor antagonist omwe amagwira ntchito poletsa zotsatira za bradykinin, mkhalapakati wofunikira wa kutupa komwe kumayenderana ndi HAE. Icatibant acetate imaperekedwa kudzera mu jakisoni wa subcutaneous ndipo idapangidwa kuti ichepetse mwachangu zizindikiro za kuukira kwa HAE koopsa.
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Ganirelix Acetate CAS: 123246-29-7
Ganirelix acetate ndi mankhwala omwe amagwiritsidwa ntchito muukadaulo wothandizira kubereka kuti apewe ovulation isanafike nthawi yobereka mwa akazi omwe akukhudzidwa ndi hyperstimulation yolamulidwa ya ovarian. Mwa kuletsa kutulutsidwa kwa luteinizing hormone, ganirelix acetate imathandiza kupewa ovulation isanakwane komanso imathandizira nthawi yoyenera yopezera mazira panthawi ya IVF. Imaperekedwa kudzera mu jakisoni wocheperako ndipo imagwira ntchito yofunika kwambiri pakuwongolera bwino chithandizo cha kusabereka.
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Linaclotide CAS: 851199-59-2
Linaclotide ndi mankhwala ochiritsira omwe amagwiritsidwa ntchito pochiza matenda a m'mimba omwe ali ndi vuto la kudzimbidwa (IBS-C) komanso kudzimbidwa kosatha. Monga agonist wa guanylate cyclase-C, linaclotide imagwira ntchito m'mimba kuti iwonjezere kutulutsa kwamadzimadzi ndikufulumizitsa kutuluka kwa matumbo, potero kuchepetsa zizindikiro monga kudzimbidwa ndi kusasangalala m'mimba.
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Ziconotide Acetate CAS: 107452-89-1
Ziconotide acetate ndi mankhwala opangidwa kuchokera ku poizoni wa nkhono ya Conus magus. Amagwiritsidwa ntchito ngati mankhwala ochepetsa ululu pochiza ululu waukulu kwa odwala omwe salola kapena sanayankhe mankhwala ena. Ziconotide acetate imaperekedwa kudzera mu infusion ya intrathecal, kupereka mpumulo kwa anthu omwe ali ndi ululu wosakhazikika.
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Degarelix CAS:214766-78-6
Degarelix ndi mankhwala oletsa gonadotropin-releasing hormone (GnRH) receptor antagonist omwe amagwiritsidwa ntchito pochiza khansa ya prostate yopita patsogolo. Imagwira ntchito poletsa kupanga testosterone mwachangu, mahomoni omwe amalimbitsa kukula kwa zotupa za prostate.
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Acetyl Octapeptide-3/1 CAS:868844-74-0
Acetyl Octapeptide-3, yomwe imadziwikanso kuti Argireline, ndi peptide yopangidwa yomwe imagwiritsidwa ntchito kwambiri muzinthu zosamalira khungu chifukwa cha mphamvu zake zoletsa ukalamba. Amakhulupirira kuti peptide iyi imagwira ntchito pochepetsa kukokana kwa minofu, zomwe zingathandize kuchepetsa mawonekedwe a mizere yopyapyala ndi makwinya, makamaka m'malo omwe mizere yowonekera imawonekera monga pamphumi ndi mozungulira maso.
