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(S)-tert-butyl 4,5,6,7-tetrahydro-1H-indazol-5-ylcarbamate CAS:955406-13-0
(S)-text{tert-butyl 4,5,6,7-tetrahydro-1H-indazol-5-ylcarbamate} ) ndi mankhwala omwe amagwiritsidwa ntchito pofufuza ndi kupanga mankhwala ngati chomangira kapena chomangira kupanga mamolekyulu omwe amagwira ntchito m'thupi. Amagwira ntchito ngati maziko ofunikira mu chemistry yamankhwala popanga mankhwala atsopano omwe amalunjika njira zinazake zamoyo kapena ma receptor.
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tert-butyl 4,5,6,7-tetrahydro-1H-indazol-5-ylcarbamate CAS:1158767-01-1
Tert-Butyl 4,5,6,7-tetrahydro-1H-indazol-5-ylcarbamate ndi mankhwala omwe amagwiritsidwa ntchito kwambiri pakufufuza ndi kupanga mankhwala ngati chinthu chothandiza kwambiri popanga mamolekyu osiyanasiyana omwe amagwira ntchito m'thupi. Mankhwalawa amagwira ntchito ngati chomangira chofunikira kwambiri mu chemistry yamankhwala, kupereka mwayi wofufuza ubale wa kapangidwe kake ndi ntchito zake ndikupanga mankhwala atsopano omwe angagwiritsidwe ntchito ndi mankhwala.
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Piperidine-2-carbonitrile hydrochloride CAS:117921-54-7
Piperidine-2-carbonitrile hydrochloride ndi mankhwala omwe amagwiritsidwa ntchito kwambiri popanga zinthu zachilengedwe komanso kafukufuku wamankhwala. Kapangidwe kake ka piperidine ndi gulu la cyano kamapereka kusinthasintha popanga mamolekyu osiyanasiyana omwe angathe kuchita zinthu zamoyo.
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4-methoxy-2,3-dihydro-1H-inden-1-ol CAS:67199-57-9
4-methoxy-2,3-dihydro-1H-inden-1-ol ndi mankhwala omwe amagwiritsidwa ntchito popanga zinthu zachilengedwe komanso mankhwala. Kapangidwe kake kapadera komwe kali ndi gulu la methoxy ndi gulu la hydroxyl kumapangitsa kuti ikhale yosangalatsa kwambiri pokonzekera mamolekyu osiyanasiyana achilengedwe omwe angakhale ndi zochita zamoyo.
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methyl isoquinoline-8-carboxylate CAS:850858-56-9
Methyl isoquinoline-8-carboxylate ndi mankhwala omwe amagwiritsidwa ntchito popanga zinthu zachilengedwe komanso kafukufuku wamankhwala. Kapangidwe kake ka isoquinoline kumapangitsa kuti ikhale chinthu chofunikira kwambiri pokonzekera mamolekyu osiyanasiyana omwe angakhale ndi zochita zamoyo.
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Tobramycin Base CAS:32986-56-4
Tobramycin base ndi mankhwala opha tizilombo toyambitsa matenda omwe amagwiritsidwa ntchito kwambiri pochiza matenda osiyanasiyana a bakiteriya, makamaka omwe amakhudza maso ndi khungu. Ndi a gulu la aminoglycoside la maantibayotiki ndipo amagwira ntchito poletsa kupanga mapuloteni a bakiteriya, zomwe zimapangitsa kuti maselo a bakiteriya afe. Tobramycin base imapezeka m'njira zosiyanasiyana, kuphatikizapo madontho a m'maso, mafuta odzola, ndi jakisoni, zomwe zimathandiza kuti igwiritsidwe ntchito m'njira zosiyanasiyana kutengera mtundu wa matenda komanso kuopsa kwake.
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trans-2-Carbomethoxycyclohexane-1-carboxyicacidCAS:2484-60-8
Trans-2-Carbomethoxycyclohexane-1-carboxyic acid ndi mankhwala omwe amagwiritsidwa ntchito popanga zinthu zachilengedwe komanso mankhwala. Kapangidwe kake kapadera komanso magulu ake ogwira ntchito zimapangitsa kuti ikhale molekyulu yosangalatsa popanga mankhwala atsopano okhala ndi zinthu zosiyanasiyana.
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Tilmicosin CAS:108050-54-0
Tilmicosin ndi mankhwala opha tizilombo omwe ali m'gulu la macrolide, omwe amagwiritsidwa ntchito kwambiri m'ziweto, makamaka m'ng'ombe ndi nkhumba. Amachiritsa bwino matenda opumira omwe amayamba chifukwa cha mabakiteriya ena, monga Pasteurella spp. ndi Mycoplasma spp. Tilmicosin imagwira ntchito poletsa kupanga mapuloteni a mabakiteriya, motero imaletsa kukula ndi kuberekana kwawo.
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Vancomycin hydrochloride CAS:1404-93-9
Vancomycin hydrochloride ndi mankhwala amphamvu opha tizilombo omwe amagwiritsidwa ntchito makamaka pochiza matenda akuluakulu a bakiteriya, makamaka omwe amayamba chifukwa cha mabakiteriya omwe ali ndi gramu omwe sagonjetsedwa ndi maantibayotiki ena. Ndi m'gulu la maantibayotiki a glycopeptide ndipo amagwira ntchito poletsa kupanga makoma a maselo a bakiteriya, zomwe zimapangitsa kuti maselo afe. Vancomycin hydrochloride nthawi zambiri imaonedwa ngati "njira yomaliza" yopha tizilombo toyambitsa matenda omwe sayankha mankhwala ena.
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Trimethoprim CAS:3380-34-5
Trimethoprim ndi mankhwala opha tizilombo toyambitsa matenda omwe amagwiritsidwa ntchito pochiza matenda osiyanasiyana a bakiteriya, makamaka omwe amakhudza njira ya mkodzo, njira yopumira, ndi khungu. Ndi m'gulu la maantibayotiki oletsa dihydrofolate reductase, omwe amagwira ntchito poletsa kupanga tetrahydrofolic acid, yomwe ndi yofunika kwambiri pakukula ndi kuberekana kwa mabakiteriya. Trimethoprim nthawi zambiri imagwiritsidwa ntchito limodzi ndi sulfamethoxazole, ndikupanga co-trimoxazole (TMP-SMX) ya mankhwala opha tizilombo toyambitsa matenda. Kuphatikiza kumeneku kumawonjezera mphamvu ya mabakiteriya ndipo kumathandiza kupewa kukula kwa kukana kwa mabakiteriya.
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Tylosin tartrate CAS: 74610-55-2
Tylosin tartrate ndi mankhwala opha tizilombo omwe amagwiritsidwa ntchito kwambiri pochiza matenda osiyanasiyana m'ziweto, makamaka nkhuku ndi nkhumba. Ndi m'gulu la ma macrolide a maantibayotiki ndipo amagwira ntchito polimbana ndi mabakiteriya okhala ndi gramu, mycoplasma, ndi ma protozoa ena. Tylosin tartrate imagwira ntchito poletsa kupanga mapuloteni a mabakiteriya, motero imasokoneza kukula ndi kuberekana kwa mabakiteriya.
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Trimethoprim CAS:738-70-5
Trimethoprim ndi mankhwala opha tizilombo toyambitsa matenda omwe amagwiritsidwa ntchito pochiza matenda osiyanasiyana a bakiteriya, makamaka omwe amakhudza njira ya mkodzo, njira yopumira, ndi khungu. Ndi m'gulu la maantibayotiki oletsa dihydrofolate reductase, omwe amagwira ntchito poletsa kupanga tetrahydrofolic acid, yomwe ndi yofunika kwambiri pakukula ndi kuberekana kwa mabakiteriya. Trimethoprim nthawi zambiri imagwiritsidwa ntchito limodzi ndi sulfamethoxazole, ndikupanga co-trimoxazole (TMP-SMX) ya mankhwala opha tizilombo toyambitsa matenda. Kuphatikiza kumeneku kumawonjezera mphamvu ya mabakiteriya ndipo kumathandiza kupewa kukula kwa kukana kwa mabakiteriya.
