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Hydrocortisone Base CAS: 50-23-7 Wopanga Wogulitsa
Hydrocortisone, 11β,17,21-trihydroxypregn-4-ene-3,20-dione, ndiye munthu wamkulu wachilengedwe wa GCin. Ngakhale kuti pali ma GC ambiri opangidwa, hydrocortisone, ma esters ake, ndi mchere wake akadali chinthu chofunikira kwambiri pa chithandizo chamakono cha adrenocortical steroid komanso muyezo woyerekeza ma GC ena onse ndi ma MC. Imagwiritsidwa ntchito pa zizindikiro zonse zomwe zatchulidwa kale.
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Orlistat CAS:96829-58-2 Wogulitsa Wopanga
Orlistat ndi mankhwala oletsa kugaya chakudya otchedwa lipase inhibitors. Orlistat idayambitsidwa ku UK ngati Xenical pochiza kunenepa kwambiri kwa nthawi yayitali, makamaka limodzi ndi zakudya zochepa zama calories. Orlistat ndi mankhwala ochokera ku lipstatin yachilengedwe ya hypolipidemic (yochokera ku Streptomyces toxyfncini) ndipo imapezeka mwa hydrogenation ya lipstatine kapena njira zosiyanasiyana zopangira zomwe zimaphatikizapo masitepe ambiri kuchokera ku (S) - rnalic acid.
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L-Homoarginine Monohydrochloride CAS:1483-01-8 Wopanga Wogulitsa
L-Homoarginine ndi mankhwala oletsa alkaline phosphatases omwe sapikisana komanso opangidwa ndi ziwalo zina. Amino acid yosafunikira iyi imaletsa mafupa ndi chiwindi cha anthu alkaline phosphatases koma siikhudza ma isoenzymes a placental kapena matumbo. Chithandizo chisanachitike ndi L-homoarginine chimachedwetsa kukula kwa chotupa m'thupi mwa mtundu wa C3H/He osteosarcoma. Imaletsanso kukula kwa pancreatic komwe kumayambitsidwa ndi mapuloteni ambiri komanso kutulutsa ma enzyme m'makoswe omwe amasinthidwa ndi madzi a bile, chitsanzo choyambitsa kutulutsa kwa pancreatic enzyme ndi hypercholecystokininemia..
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Escitalopram Oxalate CAS:219861-08-2
Escitalopram oxalate ndi metabolite ya S-isomer ya citalopram ndipo ndi gawo lalikulu la ntchito yake ya mankhwala. Dzina lake la mankhwala ndi (S) -1- [3- (dimethylamino) propyl] -1- (Chemicalbook4-fluorophenyl) -1,3-dihydroisobenzofuran 5-acetonitrile oxalate, Ndi choletsa chosankha cha serotonin reuptake, Chili ndi zotsatira zabwino zochizira kuvutika maganizo kwachibadwa komanso kosabadwa.
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Kuchepetsa Glutathione CAS: 70-18-8 Wopanga Wogulitsa
Glutathione (GSH) ndi tripeptide (γ-glutamylcysteinylglycine) yomwe imafalikira kwambiri m'zomera ndi nyama. GSH imagwira ntchito ngati nucleophilic co-substrate ku glutathione transferases pochotsa poizoni m'thupi la xenobiotics ndipo ndi wopereka ma elekitironi ofunikira ku glutathione peroxidases pochepetsa ma hydroperoxides. GSH imagwiranso ntchito poyendetsa amino acid ndikusunga kuchepa kwa mapuloteni a sulfhydryl. Kuchuluka kwa GSH kumayambira pa micromolar yochepa mu plasma mpaka millimolar ingapo m'maselo monga chiwindi.
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Cysteine CAS: 52-90-4 Wopanga Wogulitsa
L-Cysteine ndi imodzi mwa ma amino acid 20 achilengedwe ndipo, kupatula methionine, yokhayo yomwe ili ndi sulfure. Ndi amino acid yosafunikira yokhala ndi thiol yomwe imasungunuka kuti ipange Cystine. Ndi amino acid yosafunikira yokhala ndi sulfure mwa anthu, yogwirizana ndi cystine, Cysteine ndi yofunika kwambiri popanga mapuloteni, kuchotsa poizoni m'thupi, komanso ntchito zosiyanasiyana za kagayidwe kachakudya. Imapezeka mu beta-keratin, puloteni yayikulu m'misomali, pakhungu, ndi tsitsi, Cysteine ndi yofunika kwambiri popanga collagen, komanso kusinthasintha kwa khungu ndi kapangidwe kake.
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Coenzyme A asidi yaulere CAS:85-61-0
Coenzyme A yaulere asidindi cofactor yofunika kwambiri yomwe imagwira ntchito ngati gulu la acyl komanso gulu loyambitsa carbonyl pa kayendedwe ka citric acid ndi kagayidwe ka mafuta acid. Pafupifupi 4% ya ma enzyme a m'maselo amagwiritsa ntchito CoA ngati gawo lapansi. Imapangidwa kuchokera ku pantothenic acid mu njira ya masitepe 5 yomwe imafuna ATP. Gawo la pantothenate kinase la njira ya CoA biosynthetic ladziwika kuti ndi chandamale cha kupanga mankhwala oletsa mabakiteriya.
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Idebenone CAS: 58186-27-9 Wopanga Wogulitsa
Idebenone ndi mankhwala achilengedwe ochokera m'banja la quinone, ofanana ndi coenzyme Q-10. Ndi mtundu wa mankhwala opangidwa ndi Takeda Pharmaceutical Company pochiza matenda a Alzheimer's ndi zilema zina zamaganizo. Komabe, izi sizinapite patsogolo kwambiri chifukwa cha chizindikirochi. Tsopano ikugwiritsidwanso ntchito pochiza Friedreich's ataxia zomwe zimakhudza kwambiri kuthamanga kwa magazi m'thupi komanso ntchito ya mitsempha.
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Tetracaine Hydrochloride CAS:136-47-0 Wopanga Wogulitsa
Tetracaine hydrochloride ndi benzoate ester. Ndi mankhwala amphamvu oletsa ululu am'deralo a mtundu wa ester omwe amagwiritsidwa ntchito pochiza ululu pamwamba ndi msana. Tetracaine hydrochloride ndi mankhwala oletsa ululu am'deralo komanso opangidwa kuchokera ku p-amino benzoic acid. Amachita posokoneza kulowa kwa ma sodium ion m'maselo a mitsempha ndipo ndi imodzi mwa mankhwala oletsa ululu omwe amagwiritsidwa ntchito kwambiri.
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Leucine CAS: 61-90-5 Wopanga Wogulitsa
Leucine ndi imodzi mwa ma amino acid asanu ndi atatu ofunikira, ndipo ndi ya aliphatic amino acid mkati mwa mitundu makumi awiri ya mapuloteni. L-leucine ndi L-isoleucine ndi L-valine amatchedwa ma amino acid atatu okhala ndi nthambi. L-leucineLeucine ndi D-leucine ndi enantiomers. Ndi kristalo yoyera yonyezimira ya hexahedral kapena ufa woyera wa kristalo kutentha kwa chipinda, Yopanda fungo, yowawa pang'ono. Pakakhala ma hydrocarbons, imakhala yokhazikika mu asidi yamchere yamadzi. Pa gramu iliyonse imasungunuka m'madzi a 40ml ndi pafupifupi 100ml acetic acid. Imasungunuka pang'ono mu ethanol kapena ether, imasungunuka mu formic acid, imasungunuka mu hydrochloric acid, yankho la alkali hydroxides ndi yankho la carbonates.
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Guanidinopropionic Acid CAS:353-09-3 Wopanga Wogulitsa
Guanidinopropionic acid ndi kristalo woyera womwe umasungunuka m'madzi ndipo ndi creatine analog. Guanidinopropionic acid ndi mtundu wa amino acid derivatives. Ndi mankhwala ofunikira komanso ofunikira kwambiri. Amapezeka mu seramu yamagazi, ubongo, chiwindi, impso ndi mkodzo wa nyama zoyamwitsa.
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Olmesartan CAS:144689-24-7 Wogulitsa Wopanga
Olmesartan medoxomil,phenyl]phenyl]methyl]imidazole-4-carboxylate (Benicar, Olmetec) imagwiritsa ntchito tetrazolering system ngati acidity system yake, yomwe imagwira ntchito pomanga ma receptor. Ikaperekedwa kwa wodwala, mankhwalawa amayambitsidwa mwachangu komanso kwathunthu ndi ester hydrolysis ya medoxomil panthawi yoyamwa kuchokera m'mimba. Olmesartan ndi biphenylyltetrazole. Ili ndi ntchito ngati antihypertensive agent komanso angiotensin receptor antagonist.
