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Celecoxib CAS:169590-42-5 Wogulitsa Wopanga
Celecoxib ndi membala wa gulu la ma pyrazoles omwe ndi 1H-pyrazole omwe amalowetsedwa m'malo 1, 3 ndi 5 ndi magulu a 4-sulfamoylphenyl, trifluoromethyl ndi p-tolyl, motsatana. Ndi choletsa cha cyclooxygenase-2, chimagwiritsidwa ntchito pochiza nyamakazi. Chimagwira ntchito ngati choletsa cha cyclooxygenase 2, geroprotector, mankhwala oletsa kutupa osagwiritsa ntchito steroidal komanso mankhwala ochepetsa ululu osagwiritsa ntchito mankhwala osokoneza bongo. Ndi membala wa toluenes, sulfonamide, membala wa pyrazoles ndi mankhwala a organofluorine.
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Palmitoylethanolamide CAS: 544-31-0 Wopanga Wogulitsa
Palmitoylethanolamide (PEA) ndi mafuta acid amide omwe amapangidwa m'thupi omwe amamangirira ndikuyambitsa peroxisome proliferator-activated receptor alpha (PPAR-α). Poyamba idafotokozedwa ngati agonist ya mtundu wachiwiri wa cannabinoid receptor (CB2), ngakhale tsopano zadziwika kuti PEA siimangirira ku ma cannabinoid receptors. PEA imadziwika kuti ili ndi mphamvu zotsutsana ndi kutupa, kumachepetsa ululu, komanso kuteteza mitsempha. Zowonjezera za PEA zagwiritsidwa ntchito ndi anthu omwe ali ndi ululu wosatha komanso omwe ali ndi ululu wa neuropathic.
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N-Acetyl-L-Carnitine HCl CAS: 5080-50-2 Wogulitsa Wopanga
Acetyl-L-carnitine ndi mtundu wa acetylated wa L-carnitine yofunika kwambiri ya mitochondrial yomwe imasinthidwa ndi ma esterases a plasma kukhala carnitine. Acetyl-L-carnitine imathandizira kutengedwa kwa acetyl-CoA mu mitochondria panthawi ya oxidation ya mafuta acid, imawonjezera kupanga acetylcholine, komanso imalimbikitsa kupanga mapuloteni ndi phospholipid. Mu thupi, acetyl-L-carnitine (100 mg/kg) imawonjezera kuchuluka kwa mapuloteni a mGlu2/3 receptor ndi ululu wamakina mu chitsanzo cha mbewa cha ululu wopweteka wokhazikika woyambitsidwa ndi Freund’s adjuvant yonse.
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Esomeprazole Magnesium CAS:161973-10-0
Esomeprazole Magnesium, choletsa pump ya proton (PPI), ndi S-isomer ya omeprazole. Esomeprazole ili ndi zilembo zovomerezeka ndi FDA kuti zigwiritsidwe ntchito pochiza matenda a reflux a gastroesophageal (GERD), kuphatikizapo kuchiritsa ndi kusunga machiritso a erosive esophagitis komanso ngati gawo la mankhwala atatu a Helicobacter pylori.
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Ribonucleic acid kuchokera ku yisiti ya wophika mkate CAS:63231-63-0
Ribonucleic acid (RNA) ndi chinthu chomwe chimapanga filimu pamwamba chomwe chimagwira ntchito yonyowetsa. Ichi ndi polyribonucleotide yomwe imapezeka mu nyukiliyasi ndi mu cytoplasm ya maselo. Transfer RNA imachotsedwa ku yisiti ya brewer. Transfer RNA iyi ndi yapadera yotumizira amino acid phenylalanine.
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Cystine CAS: 923-32-0 Wopanga Wogulitsa
Cystine imathandiza kupanga khungu ndipo ndi yofunika kwambiri pochotsa poizoni m'thupi. Mwa kuchepetsa mphamvu ya thupi yoyamwa mkuwa, cystine imateteza maselo ku poizoni wa mkuwa. Ikasinthidwa kukhala sulfuric acid, imatulutsa sulfuric acid, ndipo sulfuric acid imalumikizana ndi zinthu zina kuti iwonjezere ntchito yochotsa poizoni m'thupi lonse.
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L-Arginine L-Glutamate CAS:4320-30-3 Wogulitsa Wopanga
L-Arginine L-Glutamatendiye wopereka nayitrogeni popanga nitric oxide.L-Arginine L-GlutamateIngagwiritsidwe ntchito pa vuto la m'mimba losagwira bwino ntchito kapena kusagwira bwino ntchito monga kafukufuku wa dyspepsia.
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Coenzyme A sodium salt hydrate CAS:55672-92-9
Coenzyme A sodium salt hydratendi chinthu chofunikira kwambiri m'zinthu zamoyo ndipo chimapangidwa kuchokera ku pantothenic acid (vitamini B5). Mlingo wa CoA mu mitochondria ndi peroxisomes umafanana ndi 2-5 mM ndi 0.7 mM, motsatana.Coenzyme A sodium salt hydratendi coenzyme yomwe imathandizira kusintha kwa ma enzyme acyl-group ndikuthandizira kupanga ndi okosijeni wa mafuta acids.
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Indometacin CAS: 53-86-1 Wopanga Wogulitsa
Indomethacin (Indocin) imagwiritsidwa ntchito pochiza matenda a gouty arthritis, rheumatoid arthritis, ankylosing spondylitis, ndi osteoarthritis. Sikoyenera kugwiritsidwa ntchito ngati mankhwala ochepetsa ululu kapena oletsa kutupa chifukwa chakuti imatha kuyambitsa poizoni. Indomethacin imagwiritsidwa ntchito pa matenda a rheumatoid arthritis, nonspecific infectious polyarthritis, gouty arthritis, osteoarthritis, ankylosing spondylitis, arthrosis, kupweteka kwa msana, neuralgia, myalgia, ndi matenda ena otsagana ndi kutupa.
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Tetraethylene Glycol CAS: 112-60-7 Wopanga Wopanga
Tetraethylene glycol ndi polima yokhala ndi mayunitsi a ethylene glycol monomer ndi magulu awiri a terminal hydroxyl. Magulu a hydroxyl amatha kuchitapo kanthu kuti awonjezere kutulutsa kwa mankhwalawa. Ma compound a ethylene glycol ali ndi mawonekedwe osangalatsa a hydrophilic. Kusungunuka kwa polima kumawonjezeka pamene chiwerengero cha magulu a ethylene glycol chikuwonjezeka.
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Isoleucine CAS: 7004-09-3 Wopanga Wogulitsa
Isoleucine (yofupikitsidwa ngati Ile kapena I) ndi α - amino acid yokhala ndi formula ya mankhwala HO2CCH(NH2)CH(CH3)CH2CH3. Ndi amino acid yofunika kwambiri, zomwe zikutanthauza kuti anthu sangathe kuipanga, kotero iyenera kumezedwa. Ma codon ake ndi AUU, AUC ndi AUA. Ndi unyolo wa hydrocarbon side, isoleucine imagawidwa ngati amino acid ya hydrophobic. Pamodzi ndi threonine, isoleucine ndi imodzi mwa ma amino acid awiri omwe ali ndi unyolo wa chiral side.
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Arachidonic Acid CAS: 506-32-1 Wopanga Wogulitsa
Arachidonic acid (AA, nthawi zina ARA) ndi mtundu wa omega-6 fatty acid yomwe imayambitsa kutupa. Monga ma omega-6 fatty acid ena, arachidonic acid ndi yofunika kwambiri pa thanzi lanu. Omega-6 fatty acids imathandiza kuti ubongo wanu ugwire ntchito bwino komanso kuti ukhale ndi mphamvu yokulira. Kudya zakudya zokhala ndi omega-6 ndi omega-3 fatty acids kumachepetsa chiopsezo chanu chokhala ndi matenda a mtima. Arachidonic acid makamaka imathandiza kuwongolera ntchito ya mitsempha.
Ufa wa Arachidonic acid umasungunuka m'madzi ndipo umapangidwa mosavuta ngati emulsion yokhazikika.
