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Zogulitsa

Olmesartan Medoxomil CAS:144689-63-4 Wogulitsa Wopanga

Olmesartan Medoxomil, ndi mankhwala atsopano osankhidwa komanso opikisana a angiotensin II type 1 receptor antagonist ndipo amaletsa mwamphamvu mayankho a Ang.ll-induced pressor. Mankhwalawa adaletsa mopikisana kumangirira kwa [125I1]-All ku ma receptor a AT1 mu membrane ya adrenal cortical ya ng'ombe, koma sanakhudze kumangirira kwa ma receptor a AT2 mu membrane ya cerebellar ya ng'ombe. Olmesartan medoxomil idawonetsedwanso kuti imachepetsa kuthamanga kwa magazi bwino kwambiri kuposa losartan ndi ACE inhibitor captopril komanso bwino ngati pbloker atenolol.


Tsatanetsatane wa Zamalonda

Ma tag a Zamalonda

Kugwiritsa Ntchito ndi Zotsatira zake

Olmesartan medoxomil ndi mankhwala oletsa angiotensin II receptor omwe amagwiritsidwa ntchito pochiza kuthamanga kwa magazi. Olmesartan imagwira ntchito poletsa kumangirira kwa angiotensin II ku ma AT1 receptors mu minofu ya mitsempha yamagazi. Mwa kuletsa kumangirira m'malo mopanga angiotensin II, olmesartan imaletsa mayankho oipa pa kutulutsidwa kwa renin m'thupi. Olmesartan medoxomil ndi mankhwala omwe amachotsedwa ku metabolite yogwira ntchito, olmesartan. Olmesartan ili ndi njira ziwiri zochotsera, ndipo pafupifupi 60% imachotsedwa ndi chiwindi ndi yotsalayo ndi impso. Pazochitika za impso kapena chiwindi chofooka, njira ina yotulutsira mankhwala imatha kulipira vuto lomwe lawonongeka.

Chitsanzo cha Zamalonda

Chithunzi cha 362(1)
Zithunzi za 320(1)

Kulongedza Zinthu:

Chithunzi 81(1)

Zina Zowonjezera:

Kapangidwe kake C29H30N6O6
Kuyesa 99%
Maonekedwe Ufa woyera mpaka beige
Nambala ya CAS 144689-63-4
Kulongedza 25KG
Moyo wa Shelufu zaka 2
Malo Osungirako Sungani pamalo ozizira komanso ouma
Chitsimikizo ISO.

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