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Rapamycin kuchokera ku Streptomyces hygroscopicus CAS:53123-88-9

Rapamycin ndi mankhwala achilengedwe omwe amapangidwa kuchokera ku bakiteriya ya Streptomyces hygroscopicus. Ili ndi ntchito zambiri zamoyo ndipo imadziwika kwambiri chifukwa cha mphamvu zake zoletsa chitetezo cha mthupi komanso zotsutsana ndi khansa.

Poyamba idapezeka ngati mankhwala opha mavairasi, rapamycin yapezeka kuti ili ndi mphamvu zoletsa chitetezo cha mthupi, zomwe zimapangitsa kuti ikhale yothandiza kwambiri poika ziwalo zina kuti isakanidwe. Imachita izi mwa kuletsa kuyambika ndi kufalikira kwa maselo a T, omwe ndi gawo lofunika kwambiri pa chitetezo cha mthupi.

Kuphatikiza apo, rapamycin yawonetsa zotsatira zabwino pochiza khansa zosiyanasiyana. Imagwira ntchito poletsa puloteni yotchedwa mTOR (chinthu chomwe chimayambitsa mammary target of rapamycin), yomwe imagwira ntchito yofunika kwambiri pakukula ndi kugawikana kwa maselo. Mwa kuletsa mTOR, rapamycin imathandiza kuwongolera kukula kosalamulirika kwa maselo a khansa.


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Kugwiritsa Ntchito ndi Zotsatira zake

Mphamvu Yosintha Thupi la Munthu: Rapamycin imaletsa kugwira ntchito ndi kuchulukana kwa maselo a T, zomwe ndizofunikira kwambiri pa chitetezo chamthupi. Mphamvu yoletsa chitetezo chamthupi imeneyi imapangitsa kuti ikhale yothandiza poika ziwalo zina kuti isakanidwe.

Ntchito Yolimbana ndi Khansa: Rapamycin yakhala ikugwira ntchito ngati mankhwala oletsa khansa. Imaletsa puloteni ya mTOR, yomwe imagwira ntchito pakukula ndi kugawikana kwa maselo. Poyang'ana mTOR, rapamycin imathandiza kuwongolera kukula kwambiri kwa maselo a khansa. Yaphunziridwa mitundu yosiyanasiyana ya khansa, kuphatikizapo khansa ya m'mawere, ya prostate, ya m'mapapo, ndi ya impso.

Kuchiza Matenda Osowa: Rapamycin yavomerezedwa kuti igwiritsidwe ntchito pochiza matenda ena osowa, monga lymphangioleiomyomatosis (LAM) ndi tuberous sclerosis complex (TSC). Matendawa amakhudza kukula kosazolowereka kwa maselo m'ziwalo zosiyanasiyana, ndipo rapamycin imathandiza kuwongolera zizindikiro ndi kupita patsogolo kwa matendawa.

Zotsatira Zoletsa Kutupa: Rapamycin yawonetsa mphamvu zoletsa kutupa. Imatha kuletsa maselo ena a chitetezo chamthupi ndi mapuloteni otupa, zomwe zingakhale zothandiza pa matenda otupa osatha, monga matenda odziteteza ku matenda a autoimmune.

Matenda a Mitsempha: Kafukufuku akusonyeza kuti rapamycin ikhoza kukhala ndi mphamvu pochiza matenda owononga mitsempha monga matenda a Alzheimer's ndi matenda a Parkinson. Yawonetsa kuti imateteza mitsempha komanso imaletsa ukalamba m'maphunziro okonzekera kuchipatala, koma kafukufuku wowonjezereka akufunika.

Kuletsa Ukalamba ndi Kukhala ndi Moyo Wautali: Rapamycin yatchuka chifukwa cha kuthekera kwake kotalikitsa moyo ndikulimbikitsa ukalamba wathanzi. Yaphunziridwa m'zamoyo zosiyanasiyana, ndipo zotsatira zake zasonyeza kuti moyo umawonjezeka komanso thanzi limakula.

Kulongedza Zinthu:

试剂包装2

Zina Zowonjezera:

Kapangidwe kake C51H79NO13
Kuyesa 99%
Maonekedwe Ufa woyera
Nambala ya CAS 53123-88-9
Kulongedza Kakang'ono komanso kochuluka
Moyo wa Shelufu zaka 2
Malo Osungirako Sungani pamalo ozizira komanso ouma
Chitsimikizo ISO.

 


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