Lamba ndi Njira: Mgwirizano, Mgwirizano ndi Kupambana-Kupambana
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Venlafaxine CAS:93413-69-5

Venlafaxine ndi mankhwala oletsa kupsinjika maganizo a gulu la serotonin ndi norepinephrine reuptake inhibitor (SNRI). Mankhwalawa adapangidwa koyamba ndi Wyeth mu 19Chemicalbook93 ndipo tsopano akugulitsidwa ndi Pfizer. Mankhwalawa avomerezedwa kuti agwiritsidwe ntchito pochiza matenda aakulu ovutika maganizo (MDD), matenda ovutika maganizo (GAD), komanso kuvutika maganizo komwe kumayenderana ndi nkhawa.


Tsatanetsatane wa Zamalonda

Ma tag a Zamalonda

Kugwiritsa Ntchito ndi Zotsatira zake

Venlafaxine imatha kuletsa kubwezeretsedwanso kwa NA ndi 5-HT, komanso kuletsa pang'ono kubwezeretsedwanso kwa dopamine. Kuletsa kwa cholinergic receptors mu vitro, histamine receptors α Ma receptors onsewa alibe mphamvu. Kuyamwa m'mimba ndi kwabwino, ndipo Chemicalbook imasinthidwa ndi cytochrome P45011D6 m'chiwindi ndikutulutsidwa ndi mkodzo. T1/2 ya metabolites yayikulu yogwira ntchito imayambira maola 5 mpaka 11. Pambuyo pa masabata atatu, kuchuluka kwa steady-state kunafikiridwa. Kugwiritsidwa ntchito pochiza kuvutika maganizo.

Chitsanzo cha Zamalonda

图片6
Chithunzi cha 314(1)

Kulongedza Zinthu:

Chithunzi cha 35

Zina Zowonjezera:

Kapangidwe kake C17H27NO2
Kuyesa 99%
Maonekedwe Ufa woyera wa kristalo
Nambala ya CAS 93413-69-5
Kulongedza 25KG
Moyo wa Shelufu zaka 2
Malo Osungirako Sungani pamalo ozizira komanso ouma
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