Lamba ndi Njira: Mgwirizano, Mgwirizano ndi Kupambana-Kupambana
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Zogulitsa

Clascoterone CAS:19608-29-8 Wopanga Wogulitsa

Clascoterone ndi mankhwala oletsa androgen receptor omwe akupangidwa ngati kirimu ndi yankho la Cassiopea (kampani yopangidwa ndi Cosmo Pharmaceuticals) pochiza matenda a khungu omwe amadalira androgen, kuphatikizapo androgenetic alopecia ndi acne vulgaris. Ngakhale kuti njira yeniyeni yomwe clascoterone imagwirira ntchito pochiza acne vulgaris sikudziwika, mankhwalawa akukhulupirira kuti amapikisana ndi androgen dihydrotestosterone pomangirira ku ma androgen receptors mu sebaceous gland ndi ma follicles a tsitsi kuti achepetse zizindikiro zofunika kuti ziphuphu ziyambe kufalikira.


Tsatanetsatane wa Zamalonda

Ma tag a Zamalonda

Kugwiritsa Ntchito ndi Zotsatira zake

Clascoterone ikupangidwa ngati kirimu wopaka pakhungu ndi Cassiopea wa matenda a pakhungu omwe amadalira androgen. Clascoterone (cortexolone 17α-propionate, CB-03-01) ndi mankhwala atsopano otsutsana ndi ma androgen receptors. Amalumikizana ndi ma androgen receptors ndi mphamvu yayikulu. Mwa kupikisana ndi ma androgens kuti amangirire ku ma androgen receptors, clascoterone imagwira ntchito poletsa ma androgen receptor signalling cascades omwe amalimbikitsa matenda a ziphuphu, monga kuchulukana kwa ma sebaceous gland, kupanga sebum yambiri, ndi njira zotupa. Mu Ogasiti 2020, FDA idavomereza clascoterone kuti ikhale mankhwala oyamba a ziphuphu (acne vulgaris) mwa odwala amuna ndi akazi azaka 12 kapena kuposerapo. Clascoterone ikufufuzidwanso ngati mankhwala atsopano a androgenetic alopecia.

Chitsanzo cha Zamalonda

Chithunzi cha 115(1)
Chithunzi cha 105(1)

Kulongedza Zinthu:

Chithunzi cha 116(1)

Zina Zowonjezera:

Kapangidwe kake C24H34O5
Kuyesa 99%
Maonekedwe Ufa woyera
Nambala ya CAS 19608-29-8
Kulongedza 25KG
Moyo wa Shelufu zaka 2
Malo Osungirako Sungani pamalo ozizira komanso ouma
Chitsimikizo ISO.

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