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5-Bromo-2-chloro-4-(cyclopentylamino)pyrimidine CAS:733039-20-8
5-Bromo-2-chloro-4-(cyclopentylamino)pyrimidine ndi mankhwala omwe amafufuzidwa mu kafukufuku wamankhwala. Ali ndi kapangidwe ka pyrimidine komwe kali ndi bromo ndi chloro m'malo mwake, komwe kungakhale kothandiza pakugwiritsa ntchito pochiza, kulunjika ku njira zinazake za matenda kapena njira zamoyo popezera mankhwala.
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4-[6-[[6-(1-Butoxyvinyl)-8-cyclopentyl-5-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino]pyridin-3-yl]piperazine-1-carboxylic acid tert-butyl ester CAS:866084-31-3
4-[6-[[6-(1-Butoxyvinyl)-8-cyclopentyl-5-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino]pyridin-3-yl]piperazine-1-carboxylic acid tert-butyl ester ndi mankhwala ovuta okhala ndi msana wa piperazine wokhala ndi magulu ogwira ntchito kuphatikiza pyridine, pyrimidine, ndi tert-butyl ester. Kapangidwe kake kamathandizira kugwiritsidwa ntchito komwe kungachitike mu mankhwala ndi kupanga mankhwala chifukwa cha mitundu yosiyanasiyana ya mankhwala.
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Bortezomib CAS:179324-69-7
Bortezomib ndi mankhwala omwe amagwiritsidwa ntchito pochiza matenda a multiple myeloma ndi mantle cell lymphoma. Ndi m'gulu la mankhwala oletsa proteasome, omwe cholinga chake ndi ma enzymes a proteolytic m'maselo kuti asokoneze ntchito yawo ndikuyambitsa apoptosis (kufa kwa maselo). Njira imeneyi imapangitsa kuti ikhale yothandiza polimbana ndi khansa zina zomwe maselo amakula mosalamulirika.
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Methyl 2-bromomethyl-3-nitrobenzoate CAS:98475-07-1
Methyl 2-bromomethyl-3-nitrobenzoate ndi mankhwala omwe ali ndi gulu la nitro pamalo a 3 ndi gulu la bromomethyl pamalo a 2 pamalo a msana wa benzoate. Amagwiritsidwa ntchito popanga zinthu zachilengedwe ngati chosinthira chosinthika, chomwe chimalola kupanga mamolekyu ovuta okhala ndi magulu enaake ogwira ntchito.
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Pemetrexed disodium INT-5 CAS:165049-28-5
Pemetrexed disodium INT-5 ndi mankhwala ochizira khansa omwe amagawidwa m'magulu a mankhwala oletsa folate chemotherapy. Amagwiritsidwa ntchito makamaka pochiza khansa zosiyanasiyana, kuphatikizapo mesothelioma, khansa ya m'mapapo yopanda maselo ang'onoang'ono, ndi khansa zinazake zofalikira.
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Pemetrexed disodium INT-4 CAS:137281-39-1
Pemetrexed disodium INT-4 ndi mankhwala oletsa folate chemotherapy omwe amagwiritsidwa ntchito mu khansa. Amagwiritsidwa ntchito pochiza khansa zosiyanasiyana, kuphatikizapo mesothelioma, khansa ya m'mapapo yopanda maselo ang'onoang'ono, ndi khansa zinazake zomwe zimafalikira m'thupi.
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Pemetrexed disodium INT-3 CAS:155405-80-4
Pemetrexed disodium INT-3 ndi mankhwala oletsa folate chemotherapy omwe amagwiritsidwa ntchito mu khansa. Amagwiritsidwa ntchito pochiza khansa zosiyanasiyana, kuphatikizapo mesothelioma, khansa ya m'mapapo yopanda maselo ang'onoang'ono, ndi khansa zinazake zomwe zimafalikira m'thupi.
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Terbinafine maziko CAS:91161-71-6
Terbinafine base ndi mankhwala ogwiritsidwa ntchito pochiza matenda a bowa. Ili m'gulu la allylamine la mankhwala opha mavairasi ndipo imadziwika kuti imagwira ntchito bwino polimbana ndi ma dermatophytes, yisiti, ndi nkhungu.
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2-Chloro-4,6-dimethoxy-1,3,5-triazine CAS:3140-73-6
2-Chloro-4,6-dimethoxy-1,3,5-triazine ndi mankhwala omwe amagwiritsidwa ntchito ngati chomangira chosiyanasiyana mu njira zopangira zinthu zachilengedwe komanso kusintha kwa mankhwala. Amakhala ndi magulu ogwira ntchito a chloro ndi methoxy omwe amamangiriridwa ku kapangidwe ka mphete ya triazine, zomwe zimathandiza kuti igwiritsidwe ntchito m'njira zosiyanasiyana zamakemikolo ndi mapangidwe azinthu zosiyanasiyana.
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2-Amino-4,5-bis(2-methoxyethoxy)benzonitrile CAS:950596-58-4
2-Amino-4,5-bis (2-methoxyethoxy)benzonitrile ndi mankhwala omwe amagwiritsidwa ntchito pofufuza zamankhwala, omwe amadziwika ndi kapangidwe ka benzonitrile komwe kali ndi amino ndi methoxyethoxy m'malo mwake, zomwe zingakhale zofunikira pa ntchito zinazake zochizira.
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(1R)-(S)-pinanediol-1-Ammonium Trifluoroacetate-3-methlbutane-1-boronate CAS:179324-87-9
(1R)-(S)-Pinanediol-1-Ammonium Trifluoroacetate-3-Methylbutane-1-Boronate ndi mankhwala omwe amadziwika ndi kapangidwe kovuta komwe kali ndi msana wa pinanediol, gulu la ammonium trifluoroacetate, ndi ntchito ya boronate ester. Amagwiritsidwa ntchito popanga zinthu zachilengedwe ngati chomangira chiral, zomwe zimathandiza kupanga mankhwala a stereospecific ndi mankhwala ophatikizana.
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Diethyl L-glutamate hydrochloride CAS:1118-89-4
Diethyl L-glutamate hydrochloride ndi mankhwala omwe amagwiritsidwa ntchito makamaka ngati mankhwala opangidwa pakati pa kafukufuku wa mankhwala ndi kapangidwe ka organic. Amachokera ku L-glutamic acid ndipo amagwira ntchito ngati choyambira popanga mankhwala osiyanasiyana ndi mankhwala omwe amagwira ntchito m'thupi.
