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Ezetimibe INT A CAS:189028-95-3
Ezetimibe INT A ndi mankhwala omwe cholinga chake ndi kuchiza hyperlipidemia, yomwe imadziwika ndi kuchuluka kwa cholesterol m'magazi. Imaletsa kuyamwa kwa cholesterol m'matumbo ndi ma sterol ena okhudzana nawo poyang'ana puloteni ya Niemann-Pick C1-like 1 (NPC1L1), motero imachepetsa kuchuluka kwa cholesterol m'magazi.
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Pramipexole CAS:104632-26-0
Pramipexole ndi mankhwala a dopamine agonist omwe amagwiritsidwa ntchito pochiza matenda a Parkinson ndi restless legs syndrome (RLS). Imagwira ntchito polimbikitsa ma dopamine receptors muubongo, motero imasintha zizindikiro za kuyenda kwa thupi mu matenda a Parkinson ndikuchepetsa kusasangalala mu RLS. Pramipexole imapezeka m'njira zonse ziwiri zotulutsidwa nthawi yomweyo komanso zotulutsidwa nthawi yayitali, zomwe zimapereka kusinthasintha kwa njira zochizira odwala.
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R-Tetrahydropapaverinehydrochloride CAS:54417-53-7
R-Tetrahydropapaverinehydrochloride ndi mankhwala omwe amagwiritsidwa ntchito kwambiri mu kafukufuku wamankhwala. Amadziwika ndi momwe angagwiritsire ntchito popanga mankhwala okhudzana ndi matenda amitsempha ndi mtima. Mankhwalawa amapangidwa ndikuphunziridwa chifukwa cha mphamvu zake zamankhwala, makamaka momwe amakhudzira minofu yosalala ya mitsempha ndi machitidwe a neurotransmitter. Ofufuza amafufuza zotsatira zake zochiritsira matenda monga kuthamanga kwa magazi ndi matenda ena amitsempha, cholinga chake ndikugwiritsa ntchito mankhwala ake kuti agwiritsidwe ntchito mtsogolo.
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4-(4-Aminophenyl)morpholin-3-one CAS:438056-69-0
4-(4-Aminophenyl)morpholin-3-one ndi mankhwala okhala ndi formula ya molekyulu C11H14N2O2. Amadziwikanso ndi dzina lake la IUPAC, 4-(4-Aminophenyl)morpholin-3-one. Mankhwalawa ali ndi mphete ya morpholine yomwe imalowetsedwa m'malo mwa gulu la aminophenyl pamalo a 4.
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3-[(2R,5S)-5-(4-Fluorophenyl)-2-[(S)-[(4-fluorophenyl(amino)]][4-[trimethylsilyl]-oxy]phenyl]methyl]-1-oxo-5-[(trimethylsily)-oxy]pentyl]-4-phenyl-(4S)-2-oxazolidinone CAS:272778-12-8
3-[(2R,5S)-5-(4-Fluorophenyl)-2-[(S)-[(4-fluorophenyl(amino)]][4-[trimethylsilyl]-oxy]phenyl]methyl]-1-oxo-5-[(trimethylsily)-oxy]pentyl]-4-phenyl-(4S)-2-oxazolidinone ndi mankhwala ovuta okhala ndi formula ya molekyulu C34H41F2N3O6Si2. Ndi chinthu chochokera ku oxazolidinone chomwe chimadziwika ndi zovuta zake komanso kugwiritsa ntchito mankhwala.
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4-hydroxythiobenzamide CAS:25984-63-8
4-Hydroxythiobenzamide ndi mankhwala omwe amadziwika ndi kapangidwe kake kamene kali ndi gulu la hydroxy lomwe limalumikizidwa ku thiobenzamide core. Amagwiritsidwa ntchito popanga zinthu zachilengedwe komanso kafukufuku wa mankhwala chifukwa cha magwiridwe ake apadera komanso momwe angagwiritsire ntchito m'magawo osiyanasiyana asayansi.
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(S)-4,5,6,7-Tetrahydro-2,6-benzothiazolediamine CAS:106092-09-5
(S)-4,5,6,7-Tetrahydro-2,6-benzothiazolediamine ndi mankhwala omwe amadziwika chifukwa cha kapangidwe kake komwe kali ndi maziko a benzothiazole ndi gulu la amine. Amaphunziridwa chifukwa cha momwe angagwiritsire ntchito kafukufuku wamankhwala ndi kapangidwe ka organic, chifukwa cha kapangidwe kake kapadera ka mamolekyu.
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Bupivacaine CAS:2180-92-9
Bupivacaine ndi mankhwala oletsa ululu omwe amagwira ntchito kwa nthawi yayitali omwe ali m'gulu la mankhwala a amide. Amagwira ntchito poletsa zizindikiro za mitsempha m'thupi, zomwe zimapangitsa kuti dzanzi kapena kutayika kwa kumverera m'dera linalake. Bupivacaine imagwiritsidwa ntchito kwambiri pochepetsa ululu panthawi ya opaleshoni, kubereka, ndi njira zina zamankhwala. Imagwiritsidwanso ntchito pochepetsa ululu pambuyo pa opaleshoni komanso pamavuto ena opweteka nthawi yayitali. Bupivacaine imaperekedwa ndi jakisoni ndipo imadziwika kuti ndi yamphamvu komanso yokhalitsa pochepetsa ululu.
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Atracurium oxalate CAS:64228-78-0
Atracurium oxalate ndi mankhwala omwe amagwiritsidwa ntchito ngati choletsa mitsempha ya mitsempha pochiza ululu. Ndi mankhwala ochokera ku atracurium besylate, omwe amapangidwa kuti azigwiritsidwa ntchito m'mitsempha panthawi ya opaleshoni kuti apangitse minofu kumasuka. Mankhwalawa amagwira ntchito molumikizana ndi ma cholinergic receptors pamalo olumikizirana mitsempha, motero amaletsa kufalikira kwa mitsempha ndikupangitsa minofu ya mafupa kufooka kwakanthawi. Atracurium oxalate imayamikiridwa chifukwa imayamba mwachangu komanso nthawi yayitali yogwira ntchito, zomwe zimapangitsa kuti ikhale yoyenera kuchita opaleshoni zosiyanasiyana zomwe zimafuna kupumula minofu moyenera.
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Ethyl 2-(4-hydroxyphenyl)-4-methylthiazole-5-carboxylate CAS:161797-99-5
Ethyl 2-(4-hydroxyphenyl)-4-methylthiazole-5-carboxylate ndi mankhwala omwe amagwiritsidwa ntchito pofufuza zamankhwala ndi kupanga zinthu zachilengedwe. Ndi a m'banja la thiazole ndipo amadziwika ndi magulu ake ogwirira ntchito a phenyl ndi ester. Mankhwalawa amaphunziridwa chifukwa cha ntchito zake zamoyo ndipo amapangidwa kuti agwiritsidwe ntchito m'njira zosiyanasiyana mu chemistry yamankhwala.
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2,6-Diamino-4,5,6,7-tetrahydrobenzothiazole CAS:104617-49-4
2,6-Diamino-4,5,6,7-tetrahydrobenzothiazole ndi mankhwala omwe amadziwika ndi kapangidwe kake komwe kali ndi maziko a benzothiazole ndi magulu awiri a amino. Amadziwika chifukwa cha kugwiritsidwa ntchito kwake kofunikira mu kafukufuku wamankhwala ndi kapangidwe ka organic, chifukwa cha kapangidwe kake kapadera ka mamolekyulu.
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4-[[(4-Fluorophenyl)imino]methyl]-phenol CAS:3382-63-6
4-[[(4-Fluorophenyl)imino]methyl]-phenol, yokhala ndi formula ya molekyulu C13H10FNO, ndi mankhwala omwe amadziwika ndi kapangidwe kake ka zonunkhira. Ili ndi mphete ya phenol yomwe imalowetsedwa m'malo mwa gulu la iminomethyl lomwe limalumikizidwa ku gawo la fluorophenyl.
